Investor Update
Basel, 2 November 2007
Significant
new data on Roche’s PEGASYS and Hepatitis C Pipeline compounds to be featured at 58th Annual AASLD Meeting
Roche
today announced that new study results for PEGASYS (peginterferon alfa-2a), the world’s leading treatment
for chronic hepatitis C virus (HCV) infection, as well as the company’s robust pipeline of hepatitis
C compounds in clinical development, will be presented at the upcoming 58th Annual Meeting of the American
Association for the Study of Liver Diseases (AASLD), also known as The Liver Meeting, in Boston, November
2-6, 2007.
The presentations will include final efficacy and safety results
from REPEAT, a major study examining retreatment with PEGASYS/COPEGUS (ribavirin) in patients whose
infection did not respond to prior treatment with Peg-Intron (peginterferon alfa-2b) and ribavirin.
Additionally, the first efficacy and safety results from a Phase IIa study with the polymerase
inhibitor R1626, as well as new data on the polymerase inhibitor R7128 (being developed in partnership
with Pharmasset), and the protease inhibitor R7227/ITMN-191 (being developed with InterMune), will be
presented.
“As the premier meeting in the science and practice of hepatology,
The Liver Meeting provides Roche with an important opportunity to demonstrate our commitment to advancing
the diagnosis and treatment of this devastating disease,” said Nick Cammack, Ph.D., Virology Disease
Biology Area Leader, Roche. “In addition to ongoing research with PEGASYS, reinforcing its status as
the leading HCV therapy, Roche is dedicated to developing new molecules that could help more patients
achieve treatment success.”
PEGASYS Highlights
- “Pegylated interferon alfa-2a plus ribavirin (RBV) in prior non-responders to pegylated interferon alfa-2b/RBV: final efficacy and safety outcomes of the REPEAT study,” D. M. Jensen et al., Monday, November 5, 3:45 p.m. - 4:00 p.m. ET (Oral Presentation No. LB4).
- “Rapid and early virological response rates are increased with 12 week 360 µg/wk peginterferon alfa-2a and standard ribavirin in HCV genotype 1 treatment naive patients: efficacy and safety analysis of the induction phase of the CHARIOT study,” S. Roberts et al., Sunday, November 4, 6:00 p.m. - 6:15 p.m. ET (Oral Presentation No. 54).
- “Prolonged Antiviral Therapy With Peginterferon to Prevent Complications of Advanced Liver Disease Associated With Hepatitis C: Results of the Hepatitis C Antiviral Long-term Treatment against Cirrhosis (HALT-C) Trial,” A. M. Di Bisceglie et al., Monday, November 5, 3:00 p.m. - 3:15 p.m. ET (Oral Presentation No. LB1).
- “Association of Pre-Treatment and On-Treatment Factors with Rapid Virologic Response in HCV Genotype 1 Infected Patients Treated with PegIFN-2a/RBV,” M. Rodriguez-Torres et al., Tuesday, November 6, 8:00 a.m. - 12:30 p.m. ET (Poster No. 1305).
- “Prophylactic Peginterferon Alfa-2a/Ribavirin vs. No Prophylaxis Following Orthotopic Liver Transplantation (OLT) for Hepatitis C: 24-Week Virologic and Safety Responses,” M. R. Charlton, et al., Sunday, Nov. 4, 3:00 p.m. – 3:15 p.m. ET (Oral Presentation No. 25).
Pipeline Highlights
- “Robust Synergistic Antiviral Effect of R1626 in Combination with Peginterferon alfa-2a (40KD), with or without Ribavirin – Interim Analysis Results of Phase 2a Study,” P. J. Pockros, et al., Tuesday, November 6, 2007, 9:00 a.m. - 9:15 a.m. ET (Oral Presentation No. 167).
- “A high barrier to resistance may contribute to the robust antiviral effect demonstrated by R1626 in HCV genotype 1-infected treatment-naive patients,” S. Le Pogam et al., Tuesday, November 6, 2007, 8:00 a.m. - 12:30 p.m. ET (Poster No. 1298).
- “Antiviral Activity, Pharmacokinetics, Safety, and Tolerability of R7128, a Novel Nucleoside HCV RNA Polymerase Inhibitor, Following Multiple, Ascending, Oral Doses in Patients with HCV Genotype 1 Infection Who have Failed Prior Interferon Therapy,” R. Reddy et al., Tuesday, November 6, 2007, 8:00 a.m. - 12:00 p.m. ET (Poster No. LB9).
- “Genotype Coverage of the HCV NS3/4A Protease Inhibitor ITMN-191 (R7227): Biochemical Data Reveals Potent Inhibition and Slow Dissociation with Genotype 1-6 Proteases,” P. Rajagopalan et al., Tuesday, November 6, 2007, 8:00 a.m. - 12:30 p.m. ET (Poster No. 1386).
About
PEGASYS
PEGASYS, in combination with COPEGUS (ribavirin), are indicated for the
treatment of adults with chronic hepatitis C who have compensated liver disease and have not previously
been treated with interferon alpha. Efficacy has been demonstrated in patients with compensated
liver disease and histological evidence of cirrhosis (Child-Pugh class A) and patients with HIV disease
that are clinically stable (e.g., antiretroviral therapy not required or receiving stable antiretroviral
therapy). In addition, PEGASYS in combination with COPEGUS is the first and only FDA-approved regimen
for the treatment of chronic hepatitis C in patients coinfected with
hepatitis C and
HIV. PEGASYS is the only pegylated interferon indicated for the treatment of adult patients with chronic
hepatitis B (HBeAg positive and HBeAg negative chronic hepatitis B who have compensated liver disease
and evidence of viral replication and liver inflammation).
PEGASYS is dosed at 180mcg
as a subcutaneous injection taken once a week. COPEGUS is available as a 200mg tablet, and is administered
orally two times a day as a split dose. Roche has backed PEGASYS with the most extensive clinical research
program ever undertaken in hepatitis C, with major studies initiated to advance treatment for hepatitis
C patients with unmet needs, including patients co-infected with HIV and HCV, African Americans, patients
with cirrhosis, and patients who have failed to respond to previous therapy.
About
Roche
Headquartered in Basel, Switzerland, Roche is one of the world’s leading
research-focused healthcare groups in the fields of pharmaceuticals and diagnostics. As the world’s
biggest biotech company and an innovator of products and services for the early detection, prevention,
diagnosis and treatment of diseases, the Group contributes on a broad range of fronts to improving people’s
health and quality of life. Roche is the world leader in in-vitro diagnostics and drugs for cancer and
transplantation, a market leader in virology and active in other major therapeutic areas such as autoimmune
diseases, inflammation, metabolic disorders and diseases of the central nervous system. In 2006 sales
by the Pharmaceuticals Division totalled 33.3 billion Swiss francs, and the Diagnostics Division posted
sales of 8.7 billion Swiss francs. Roche has R&D agreements and strategic alliances with numerous
partners, including majority ownership interests in Genentech and Chugai, and invests approximately
7 billion Swiss francs a year in R&D. Worldwide, the Group employs about 75,000 people. Additional
information is available on the Internet at www.roche.com.
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